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Novel Diazole/Triazole and Dibenzothiophene Dioxide Containing Pentacyclic Systems with Promising Biological Activities
Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
- 1 Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
- 2 Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
- 3 Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
- 4 Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
- 5 Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
- 6 Department of Chemical and Biological Technology, Georgian Technical University, Tbilisi, Georgia
International Journal of Organic Chemistry·Volume 07 (2016)·Pages 34–41·Published 27 December 2016·DOI10.4236/ijoc.2017.71004
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Abstract
The aim of the current work is to synthesize the new heterocyclic pentacyclic condensed systems that combine benzothiophen and benzimidazole/triazole into one molecule. The dibenzothiophene was taken as an initial compound and by consistent “extension” was annihilated the imidazole and triazole nucleuses. As a result two new pentacyclic systems were produced: 3H-, 7H-diimidazole[4,5-b][5,4-g] dibenzothiophene-5,5-dioxide and 3H-, 7H-ditriazole[4,5-b][5,4-g] dibenzothiophene-5,5-dioxide with the promising antimi-crobial activity. Their spectral characteristics were studied.
KeywordsDibenzothiophene DioxideImidazoleTriazolePentacyclic Systems
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